DPP8 Selective Inhibitor Tominostat as a Novel and Broad-Spectrum Anticancer Agent against Hematolog...
DPP8 Selective Inhibitor Tominostat as a Novel and Broad-Spectrum Anticancer Agent against Hematological Malignancies
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Author / Creator
Kikuchi, Shohei , Wada, Akinori , Kamihara, Yusuke , Okazaki, Kosuke , Jawaid, Paras , Rehman, Mati Ur , Kobayashi, Eiji , Susukida, Takeshi , Minemura, Tomoki , Nabe, Yoshimi , Iwao, Noriaki , Ozawa, Tatsuhiko , Hatano, Ryo , Yamada, Mitsugu , Kishi, Hiroyuki , Matsuya, Yuji , Mizuguchi, Mineyuki , Hayakawa, Yoshihiro , Dang, Nam H. , Sakamoto, Yasumitsu , Morimoto, Chikao and Sato, Tsutomu
Publisher
Switzerland: MDPI AG
Journal title
Language
English
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Publication information
Publisher
Switzerland: MDPI AG
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More information
Scope and Contents
Contents
DPP8/9 inhibition induces either pyroptotic or apoptotic cell death in hematological malignancies. We previously reported that treatment with the DPP8/9 inhibitor 1G244 resulted in apoptotic cell death in myeloma, and our current study further evaluates the mechanism of action of 1G244 in different blood cancer cell lines. Specifically, 1G244 inhib...
Alternative Titles
Full title
DPP8 Selective Inhibitor Tominostat as a Novel and Broad-Spectrum Anticancer Agent against Hematological Malignancies
Authors, Artists and Contributors
Author / Creator
Wada, Akinori
Kamihara, Yusuke
Okazaki, Kosuke
Jawaid, Paras
Rehman, Mati Ur
Kobayashi, Eiji
Susukida, Takeshi
Minemura, Tomoki
Nabe, Yoshimi
Iwao, Noriaki
Ozawa, Tatsuhiko
Hatano, Ryo
Yamada, Mitsugu
Kishi, Hiroyuki
Matsuya, Yuji
Mizuguchi, Mineyuki
Hayakawa, Yoshihiro
Dang, Nam H.
Sakamoto, Yasumitsu
Morimoto, Chikao
Sato, Tsutomu
Identifiers
Primary Identifiers
Record Identifier
TN_cdi_doaj_primary_oai_doaj_org_article_97715b8185fb4d6d8d5fbfbf732d6cff
Permalink
https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_doaj_primary_oai_doaj_org_article_97715b8185fb4d6d8d5fbfbf732d6cff
Other Identifiers
ISSN
2073-4409
E-ISSN
2073-4409
DOI
10.3390/cells12071100