Deactivatable Bisubstrate Inhibitors of Protein Kinases
Deactivatable Bisubstrate Inhibitors of Protein Kinases
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Publisher
Basel: MDPI AG
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Language
English
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Basel: MDPI AG
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Contents
Bivalent ligands, including bisubstrate inhibitors, are conjugates of pharmacophores, which simultaneously target two binding sites of the biomolecule. Such structures offer attainable means for the development of compounds whose ability to bind to the biological target could be modulated by an external trigger. In the present work, two deactivatab...
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Full title
Deactivatable Bisubstrate Inhibitors of Protein Kinases
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TN_cdi_doaj_primary_oai_doaj_org_article_b9b4e24415b14c1c81cc5631f9e55a9a
Permalink
https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_doaj_primary_oai_doaj_org_article_b9b4e24415b14c1c81cc5631f9e55a9a
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ISSN
1420-3049
E-ISSN
1420-3049
DOI
10.3390/molecules27196689
