Synthesis of Bispidine-Based Prostate-Specific Membrane Antigen-Targeted Conjugate and Initial Inves...
Synthesis of Bispidine-Based Prostate-Specific Membrane Antigen-Targeted Conjugate and Initial Investigations
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Author / Creator
Machulkin, Aleksei E , Petrov, Stanislav A , Kraynova, Maria D , Garanina, Anastasiia S , Egorova, Bayirta V , Timoshenko, Roman V , Vaneev, Alexander N , Erofeev, Alexander S , Priselkova, Anna B , Kalinin, Mikhail A , Aleksei V Medved′ko , Kalmykov, Stepan N , Beloglazkina, Elena K and Vatsadze, Sergey Z
Publisher
Leuven: MDPI AG
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Language
English
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Publisher
Leuven: MDPI AG
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Contents
Nowadays, PSMA ligands are widely used for radiotheragnostic purposes in prostate cancer. The synthesis of a PSMA-Bisp conjugate was developed and realized with good yield (overall yield ~58% for the last two steps). All newly synthesized compounds were characterized by physicochemical methods: 1H and 13C NMR, HRMS, and LCMS (for biologically teste...
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Full title
Synthesis of Bispidine-Based Prostate-Specific Membrane Antigen-Targeted Conjugate and Initial Investigations
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TN_cdi_doaj_primary_oai_doaj_org_article_f0413df51cf94c74bfe853d692c2c152
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https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_doaj_primary_oai_doaj_org_article_f0413df51cf94c74bfe853d692c2c152
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ISSN
2673-401X
E-ISSN
2673-401X
DOI
10.3390/org6010007
