Structure Activity Relationship and Molecular Docking of Some Quinazolines Bearing Sulfamerazine Moi...
Structure Activity Relationship and Molecular Docking of Some Quinazolines Bearing Sulfamerazine Moiety as New 3CLpro, cPLA2, sPLA2 Inhibitors
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Basel: MDPI AG
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English
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Basel: MDPI AG
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The current work was conducted to synthesize several novel anti-inflammatory quinazolines having sulfamerazine moieties as new 3CLpro, cPLA2, and sPLA2 inhibitors. The thioureido derivative 3 was formed when compound 2 was treated with sulfamerazine. Also, compound 3 was reacted with NH2-NH2 in ethanol to produce the N-aminoquinazoline derivative....
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Structure Activity Relationship and Molecular Docking of Some Quinazolines Bearing Sulfamerazine Moiety as New 3CLpro, cPLA2, sPLA2 Inhibitors
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TN_cdi_doaj_primary_oai_doaj_org_article_f8463908097e40f680939308612b4ebc
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https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_doaj_primary_oai_doaj_org_article_f8463908097e40f680939308612b4ebc
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1420-3049
E-ISSN
1420-3049
DOI
10.3390/molecules28166052