Identification of Selective ERRγ Inverse Agonists
Identification of Selective ERRγ Inverse Agonists
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Publisher
Switzerland: MDPI
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Language
English
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Publisher
Switzerland: MDPI
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Contents
GSK5182 (4) is currently one of the lead compounds for the development of estrogen-related receptor gamma (ERRγ) inverse agonists. Here, we report the design, synthesis, pharmacological and in vitro absorption, distribution, metabolism, excretion, toxicity (ADMET) properties of a series of compounds related to 4. Starting from 4, a series of analog...
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Full title
Identification of Selective ERRγ Inverse Agonists
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TN_cdi_doaj_primary_oai_doaj_org_article_51d474224d844cfc9eb9d3b1036ceb23
Permalink
https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_doaj_primary_oai_doaj_org_article_51d474224d844cfc9eb9d3b1036ceb23
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ISSN
1420-3049
E-ISSN
1420-3049
DOI
10.3390/molecules21010080
