Progress towards a public chemogenomic set for protein kinases and a call for contributions
Progress towards a public chemogenomic set for protein kinases and a call for contributions
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Author / Creator
Drewry, David H. , Wells, Carrow I. , Andrews, David M. , Angell, Richard , Al-Ali, Hassan , Axtman, Alison D. , Capuzzi, Stephen J. , Elkins, Jonathan M. , Ettmayer, Peter , Frederiksen, Mathias , Gileadi, Opher , Gray, Nathanael , Hooper, Alice , Knapp, Stefan , Laufer, Stefan , Luecking, Ulrich , Michaelides, Michael , Müller, Susanne , Muratov, Eugene , Denny, R. Aldrin , Saikatendu, Kumar S. , Treiber, Daniel K. , Zuercher, William J. and Willson, Timothy M.
Publisher
United States: Public Library of Science
Journal title
Language
English
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Publication information
Publisher
United States: Public Library of Science
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Scope and Contents
Contents
Protein kinases are highly tractable targets for drug discovery. However, the biological function and therapeutic potential of the majority of the 500+ human protein kinases remains unknown. We have developed physical and virtual collections of small molecule inhibitors, which we call chemogenomic sets, that are designed to inhibit the catalytic fu...
Alternative Titles
Full title
Progress towards a public chemogenomic set for protein kinases and a call for contributions
Authors, Artists and Contributors
Author / Creator
Wells, Carrow I.
Andrews, David M.
Angell, Richard
Al-Ali, Hassan
Axtman, Alison D.
Capuzzi, Stephen J.
Elkins, Jonathan M.
Ettmayer, Peter
Frederiksen, Mathias
Gileadi, Opher
Gray, Nathanael
Hooper, Alice
Knapp, Stefan
Laufer, Stefan
Luecking, Ulrich
Michaelides, Michael
Müller, Susanne
Muratov, Eugene
Denny, R. Aldrin
Saikatendu, Kumar S.
Treiber, Daniel K.
Zuercher, William J.
Willson, Timothy M.
Identifiers
Primary Identifiers
Record Identifier
TN_cdi_plos_journals_1926447620
Permalink
https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_plos_journals_1926447620
Other Identifiers
ISSN
1932-6203
E-ISSN
1932-6203
DOI
10.1371/journal.pone.0181585
