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Identification of Selective ERR[gamma] Inverse Agonists

Identification of Selective ERR[gamma] Inverse Agonists

https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_proquest_journals_1768909452

Identification of Selective ERR[gamma] Inverse Agonists

About this item

Full title

Identification of Selective ERR[gamma] Inverse Agonists

Publisher

Basel: MDPI AG

Journal title

Molecules (Basel, Switzerland), 2016-01, Vol.21 (1), p.80

Language

English

Formats

Publication information

Publisher

Basel: MDPI AG

More information

Scope and Contents

Contents

GSK5182 (4) is currently one of the lead compounds for the development of estrogen-related receptor gamma (ERR[gamma]) inverse agonists. Here, we report the design, synthesis, pharmacological and in vitro absorption, distribution, metabolism, excretion, toxicity (ADMET) properties of a series of compounds related to 4. Starting from 4, a series of...

Alternative Titles

Full title

Identification of Selective ERR[gamma] Inverse Agonists

Identifiers

Primary Identifiers

Record Identifier

TN_cdi_proquest_journals_1768909452

Permalink

https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_proquest_journals_1768909452

Other Identifiers

E-ISSN

1420-3049

DOI

10.3390/molecules21010080

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