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Quantitative Evaluation of mMate1 Function Based on Minimally Invasive Measurement of Tissue Concent...

Quantitative Evaluation of mMate1 Function Based on Minimally Invasive Measurement of Tissue Concent...

https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_proquest_miscellaneous_1693729750

Quantitative Evaluation of mMate1 Function Based on Minimally Invasive Measurement of Tissue Concentration Using PET with [11C]Metformin in Mouse

About this item

Full title

Quantitative Evaluation of mMate1 Function Based on Minimally Invasive Measurement of Tissue Concentration Using PET with [11C]Metformin in Mouse

Publisher

New York: Springer US

Journal title

Pharmaceutical research, 2015-08, Vol.32 (8), p.2538-2547

Language

English

Formats

Publication information

Publisher

New York: Springer US

More information

Scope and Contents

Contents

Purpose
To evaluate the function of multidrug and toxin extrusion proteins (MATEs) using
11
C-labeled metformin ([
11
C]metformin) by positron emission tomography (PET).
Methods
PET was performed by intravenous bolus injection of [
11
C]metformin. Pyrimethamine at 0.5 and 5 mg/kg was intravenously administered to mice 30...

Alternative Titles

Full title

Quantitative Evaluation of mMate1 Function Based on Minimally Invasive Measurement of Tissue Concentration Using PET with [11C]Metformin in Mouse

Identifiers

Primary Identifiers

Record Identifier

TN_cdi_proquest_miscellaneous_1693729750

Permalink

https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_proquest_miscellaneous_1693729750

Other Identifiers

ISSN

0724-8741

E-ISSN

1573-904X

DOI

10.1007/s11095-015-1642-1

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