Chemical probes to potently and selectively inhibit endocannabinoid cellular reuptake
Chemical probes to potently and selectively inhibit endocannabinoid cellular reuptake
About this item
Full title
Author / Creator
Chicca, Andrea , Nicolussi, Simon , Bartholomäus, Ruben , Blunder, Martina , Rey, Alejandro Aparisi , Petrucci, Vanessa , del Carmen Reynoso-Moreno, Ines , Viveros-Paredes, Juan Manuel , Gens, Marianela Dalghi , Lutz, Beat , Schiöth, Helgi B. , Soeberdt, Michael , Abels, Christoph , Charles, Roch-Philippe , Altmann, Karl-Heinz and Gertsch, Jürg
Publisher
United States: National Academy of Sciences
Journal title
Language
English
Formats
Publication information
Publisher
United States: National Academy of Sciences
Subjects
More information
Scope and Contents
Contents
The extracellular effects of the endocannabinoids anandamide and 2-arachidonoyl glycerol are terminated by enzymatic hydrolysis after crossing cellular membranes by facilitated diffusion. The lack of potent and selective inhibitors for endocannabinoid transport has prevented the molecular characterization of this process, thus hindering its biochem...
Alternative Titles
Full title
Chemical probes to potently and selectively inhibit endocannabinoid cellular reuptake
Authors, Artists and Contributors
Author / Creator
Nicolussi, Simon
Bartholomäus, Ruben
Blunder, Martina
Rey, Alejandro Aparisi
Petrucci, Vanessa
del Carmen Reynoso-Moreno, Ines
Viveros-Paredes, Juan Manuel
Gens, Marianela Dalghi
Lutz, Beat
Schiöth, Helgi B.
Soeberdt, Michael
Abels, Christoph
Charles, Roch-Philippe
Altmann, Karl-Heinz
Gertsch, Jürg
Identifiers
Primary Identifiers
Record Identifier
TN_cdi_swepub_primary_oai_DiVA_org_uu_329659
Permalink
https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_swepub_primary_oai_DiVA_org_uu_329659
Other Identifiers
ISSN
0027-8424,1091-6490
E-ISSN
1091-6490
DOI
10.1073/pnas.1704065114
