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Inhibition of SARS-CoV-2 main protease by allosteric drug-binding

Inhibition of SARS-CoV-2 main protease by allosteric drug-binding

https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_proquest_journals_2507152892

Inhibition of SARS-CoV-2 main protease by allosteric drug-binding

About this item

Full title

Inhibition of SARS-CoV-2 main protease by allosteric drug-binding

Author / Creator

Günther, Sebastian , Reinke, Patrick Y A , Fernández-García, Yaiza , Lieske, Julia , Lane, Thomas J , Koua, Faisal H M , Ehrt, Christiane , Ewert, Wiebke , Oberthuer, Dominik , Yefanov, Oleksandr , Meier, Susanne , Lorenzen, Kristina , Krichel, Boris , Janine-Denise Kopicki , Gelisio, Luca , Brehm, Wolfgang , Dunkel, Ilona , Seychell, Brandon , Gieseler, Henry , Norton-Baker, Brenna , Escudero-Pérez, Beatriz , Domaracky, Martin , Saouane, Sofiane , Tolstikova, Alexandra , White, Thomas A , Hänle, Anna , Groessler, Michael , Fleckenstein, Holger , Trost, Fabian , Galchenkova, Marina , Gevorkov, Yaroslav , Li, Chufeng , Awel, Salah , Peck, Ariana , Barthelmess, Miriam , Schlünzen, Frank , Xavier, P Lourdu , Werner, Nadine , Ullah, Najeeb , Falke, Sven , Srinivasan, Vasundara , Bruno Alves Franca , Schwinzer, Martin , Brognaro, Hévila , Rogers, Cromarte , Melo, Diogo , Zaitsev-Doyle, Jo J , Knoska, Juraj , Peña Murillo, Gisel E , Aida Rahmani Mashhour , Guicking, Filip , Hennicke, Vincent , Fischer, Pontus , Hakanpää, Johanna , Meyer, Jan , Gribbon, Phil , Ellinger, Bernhard , Kuzikov, Maria , Wolf, Markus , Beccari, Andrea R , Bourenkov, Gleb , David Von Stetten , Pompidor, Guillaume , Bento, Isabel , Panneerselvam, Saravanan , Karpics, Ivars , Schneider, Thomas R , Garcia Alai, Maria Marta , Niebling, Stephan , Günther, Christian , Schmidt, Christina , Schubert, Robin , Han, Huijong , Boger, Juliane , Monteiro, Diana C F , Zhang, Linlin , Sun, Xinyuanyuan , Pletzer-Zelgert, Jonathan , Wollenhaupt, Jan , Feiler, Christian G , Weiss, Manfred S , Schulz, Eike-Christian , Mehrabi, Pedram , Karničar, Katarina , Usenik, Aleksandra , Loboda, Jure , Tidow, Henning , Chari, Ashwin , Hilgenfeld, Rolf , Uetrecht, Charlotte , Cox, Russell , Beck, Tobias , Rarey, Matthias , Günther, Stephan , Turk, Dusan , Hinrichs, Winfried , Chapman, Henry N , Pearson, Arwen R , Betzel, Christian and Meents, Alke

Publisher

Cold Spring Harbor: Cold Spring Harbor Laboratory Press

Journal title

bioRxiv, 2020-11

Language

English

Formats

Publication information

Publisher

Cold Spring Harbor: Cold Spring Harbor Laboratory Press

More information

Scope and Contents

Contents

Abstract The coronavirus disease (COVID-19) caused by SARS-CoV-2 is creating tremendous health problems and economical challenges for mankind. To date, no effective drug is available to directly treat the disease and prevent virus spreading. In a search for a drug against COVID-19, we have performed a massive X-ray crystallographic screen of two re...

Alternative Titles

Full title

Inhibition of SARS-CoV-2 main protease by allosteric drug-binding

Authors, Artists and Contributors

Author / Creator

Günther, Sebastian
Reinke, Patrick Y A
Fernández-García, Yaiza
Lieske, Julia
Lane, Thomas J
Koua, Faisal H M
Ehrt, Christiane
Ewert, Wiebke
Oberthuer, Dominik
Yefanov, Oleksandr
Meier, Susanne
Lorenzen, Kristina
Krichel, Boris
Janine-Denise Kopicki
Gelisio, Luca
Brehm, Wolfgang
Dunkel, Ilona
Seychell, Brandon
Gieseler, Henry
Norton-Baker, Brenna
Escudero-Pérez, Beatriz
Domaracky, Martin
Saouane, Sofiane
Tolstikova, Alexandra
White, Thomas A
Hänle, Anna
Groessler, Michael
Fleckenstein, Holger
Trost, Fabian
Galchenkova, Marina
Gevorkov, Yaroslav
Li, Chufeng
Awel, Salah
Peck, Ariana
Barthelmess, Miriam
Schlünzen, Frank
Xavier, P Lourdu
Werner, Nadine
Ullah, Najeeb
Falke, Sven
Srinivasan, Vasundara
Bruno Alves Franca
Schwinzer, Martin
Brognaro, Hévila
Rogers, Cromarte
Melo, Diogo
Zaitsev-Doyle, Jo J
Knoska, Juraj
Peña Murillo, Gisel E
Aida Rahmani Mashhour
Guicking, Filip
Hennicke, Vincent
Fischer, Pontus
Hakanpää, Johanna
Meyer, Jan
Gribbon, Phil
Ellinger, Bernhard
Kuzikov, Maria
Wolf, Markus
Beccari, Andrea R
Bourenkov, Gleb
David Von Stetten
Pompidor, Guillaume
Bento, Isabel
Panneerselvam, Saravanan
Karpics, Ivars
Schneider, Thomas R
Garcia Alai, Maria Marta
Niebling, Stephan
Günther, Christian
Schmidt, Christina
Schubert, Robin
Han, Huijong
Boger, Juliane
Monteiro, Diana C F
Zhang, Linlin
Sun, Xinyuanyuan
Pletzer-Zelgert, Jonathan
Wollenhaupt, Jan
Feiler, Christian G
Weiss, Manfred S
Schulz, Eike-Christian
Mehrabi, Pedram
Karničar, Katarina
Usenik, Aleksandra
Loboda, Jure
Tidow, Henning
Chari, Ashwin
Hilgenfeld, Rolf
Uetrecht, Charlotte
Cox, Russell
Beck, Tobias
Rarey, Matthias
Günther, Stephan
Turk, Dusan
Hinrichs, Winfried
Chapman, Henry N
Pearson, Arwen R
Betzel, Christian
Meents, Alke

Identifiers

Primary Identifiers

Record Identifier

TN_cdi_proquest_journals_2507152892

Permalink

https://devfeature-collection.sl.nsw.gov.au/record/TN_cdi_proquest_journals_2507152892

Other Identifiers

E-ISSN

2692-8205

DOI

10.1101/2020.11.12.378422