Search the collection

2,731 results for Inverse+agonists

Sort by:

Sort by

Limit results to:

20 per page

2,731 results for Inverse+agonists

Export to excel

Export record to excel

File type to download

Beta version

Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 1
ArticlesPeer ReviewedFull Text
Advanced fluorescence microscopy reveals disruption of dynamic CXCR4 dimerization by subpocket-specific inverse agonists
Author / Creator:Işbilir, Ali ; Möller, Jan ; Arimont, Marta ; Bobkov, Vladimir ; Perpiñá-Viciano, Cristina ; Hoffmann, Carsten ; Inoue, Asuka ; Heukers, Raimond ; de Graaf, Chris ; Smit, Martine J. ; Annibale, Paolo ; Lohse, Martin J.
Publisher:United States: National Academy of Sciences
Journal title:Proceedings of the National Academy of Sciences - PNAS, 2020-11, Vol.117 (46), p.29144-29154
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 2
ArticlesPeer ReviewedFull Text
RO4938581, a novel cognitive enhancer acting at GABAA α5 subunit-containing receptors
Author / Creator:Ballard, Theresa M. ; Knoflach, Frédéric ; Prinssen, Eric ; Borroni, Edilio ; Vivian, Jeffrey A. ; Basile, Jennifer ; Gasser, Rodolfo ; Moreau, Jean-Luc ; Wettstein, Joseph G. ; Buettelmann, Bernd ; Knust, Henner ; Thomas, Andrew W. ; Trube, Gerhard ; Hernandez, Maria-Clemencia
Journal title:Psychopharmacology, 2009-01, Vol.202 (1-3), p.207-223
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 3
ArticlesPeer ReviewedFull Text
RORγt inverse agonists demonstrating a margin between inhibition of IL-17A and thymocyte apoptosis
Author / Creator:Collins, Mia ; Pehrson, Rikard ; Grindebacke, Hanna ; Leffler, Agnes ; Ramnegård, Marie ; Rannikmäe, Helena ; Krutrök, Nina ; Yrlid, Linda ; Pollard, Charlotte ; Dainty, Ian ; Narjes, Frank ; von Berg, Stefan ; Llinas, Antonio ; Malmberg, Anna ; McPheat, Jane ; Hansson, Eva ; Bäck, Elisabeth ; Bernström, Jenny ; Hansson, Thomas G. ; Keeling, David ; Jirholt, Johan
Publisher:United States: Public Library of Science
Journal title:PloS one, 2025-01, Vol.20 (1), p.e0317090
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 4
ArticlesPeer ReviewedFull Text
Structural mechanism of CB1R binding to peripheral and biased inverse agonists
Author / Creator:Kumari, Punita ; Dvorácskó, Szabolcs ; Enos, Michael D. ; Ramesh, Karthik ; Lim, Darrix ; Hassan, Sergio A. ; Kunos, George ; Cinar, Resat ; Iyer, Malliga R. ; Rosenbaum, Daniel M.
Publisher:London: Nature Publishing Group UK
Journal title:Nature communications, 2024-12, Vol.15 (1), p.10694-13, Article 10694
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 5
ArticlesPeer ReviewedFull Text
β-Arrestin-Mediated Activation of MAPK by Inverse Agonists Reveals Distinct Active Conformations for G Protein-Coupled Receptors
Author / Creator:Azzi, Mounia ; Charest, Pascale G. ; Angers, Stéphane ; Rousseau, Guy ; Kohout, Trudy ; Bouvier, Michel ; Piñeyro, Graciela
Publisher:United States: National Academy of Sciences
Journal title:Proceedings of the National Academy of Sciences - PNAS, 2003-09, Vol.100 (20), p.11406-11411
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 6
ArticlesPeer ReviewedFull Text
ROR[gamma]t inverse agonists demonstrating a margin between inhibition of IL-17A and thymocyte apoptosis
Author / Creator:Collins, Mia ; Pehrson, Rikard ; Grindebacke, Hanna ; Leffler, Agnes ; Ramnegård, Marie ; Rannikmäe, Helena ; Krutrök, Nina ; Yrlid, Linda ; Pollard, Charlotte ; Dainty, Ian ; Narjes, Frank ; von Berg, Stefan ; Llinas, Antonio ; Malmberg, Anna ; McPheat, Jane ; Hansson, Eva ; Bäck, Elisabeth ; Bernström, Jenny ; Hansson, Thomas G ; Keeling, David ; Jirholt, Johan
Publisher:Public Library of Science
Journal title:PloS one, 2025-01, Vol.20 (1), p.e0317090
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 7
ArticlesPeer ReviewedFull Text
Targeting Oxidative Stress: Novel Coumarin-Based Inverse Agonists of GPR55
Author / Creator:Apweiler, Matthias ; Saliba, Soraya Wilke ; Streyczek, Jana ; Hurrle, Thomas ; Gräßle, Simone ; Bräse, Stefan ; Fiebich, Bernd L.
Publisher:Switzerland: MDPI AG
Journal title:International journal of molecular sciences, 2021-10, Vol.22 (21), p.11665
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 8
ArticlesPeer ReviewedFull Text
Identification of Selective ERRγ Inverse Agonists
Author / Creator:Kim, Jina ; Im, Chun ; Yoo, Eun ; Ma, Min ; Kim, Sang-Bum ; Hong, Eunmi ; Chin, Jungwook ; Hwang, Hayoung ; Lee, Sungwoo ; Kim, Nam ; Jeon, Jae-Han ; Lee, In-Kyu ; Jeon, Yong ; Choi, Hueng-Sik ; Kim, Seong ; Cho, Sung
Publisher:Switzerland: MDPI
Journal title:Molecules (Basel, Switzerland), 2016-01, Vol.21 (1), p.80
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 9
ArticlesPeer ReviewedFull Text
Identification of Selective ERR[gamma] Inverse Agonists
Author / Creator:Kim, Jina ; Im, Chun Young ; Yoo, Eun Kyung ; Ma, Min Jung ; Kim, Sang-Bum ; Hong, Eunmi ; Chin, Jungwook ; Hwang, Hayoung ; Lee, Sungwoo ; Kim, Nam Doo ; Jeon, Jae-Han ; Lee, In-Kyu ; Jeon, Yong Hyun ; Choi, Hueng-Sik ; Kim, Seong Heon ; Cho, Sung Jin
Publisher:Basel: MDPI AG
Journal title:Molecules (Basel, Switzerland), 2016-01, Vol.21 (1), p.80
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 10
ArticlesPeer ReviewedFull Text
Towards Translation of PqsR Inverse Agonists: From In Vitro Efficacy Optimization to In Vivo Proof‐of‐Principle
Author / Creator:Hamed, Mostafa M. ; Abdelsamie, Ahmed S. ; Rox, Katharina ; Schütz, Christian ; Kany, Andreas M. ; Röhrig, Teresa ; Schmelz, Stefan ; Blankenfeldt, Wulf ; Arce‐Rodriguez, Alejandro ; Borrero‐de Acuña, José Manuel ; Jahn, Dieter ; Rademacher, Jessica ; Ringshausen, Felix C. ; Cramer, Nina ; Tümmler, Burkhard ; Hirsch, Anna K. H. ; Hartmann, Rolf W. ; Empting, Martin
Publisher:Germany: John Wiley & Sons, Inc
Journal title:Advanced science, 2023-02, Vol.10 (5), p.e2204443-n/a
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 11
ArticlesPeer ReviewedFull Text
The discovery of a novel series of potential ERRα inverse agonists based on p-nitrobenzenesulfonamide template for triple-negative breast cancer in vivo
Author / Creator:Gao, Zhipei ; Wang, Tianxiao ; Li, Rui ; Du, Yongli ; Lv, Han ; Zhang, Liudi ; Chen, Haifei ; Shi, Xiaojin ; Li, Qunyi ; Shen, Jingkang
Publisher:England: Taylor & Francis
Journal title:Journal of enzyme inhibition and medicinal chemistry, 2022-12, Vol.37 (1), p.125-134
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 12
ArticlesPeer ReviewedFull Text
Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (RORγt) modulators: insights into different protein behaviors with “short” and “long” inverse agonists
Author / Creator:Yu, Ming-cheng ; Yang, Feng ; Ding, Xiao-yu ; Sun, Nan-nan ; Jiang, Zheng-yuan ; Huang, Ya-fei ; Yan, Yu-rong ; Zhu, Chen ; Xie, Qiong ; Chen, Zhi-feng ; Guo, Si-qi ; Jiang, Hua-liang ; Chen, Kai-xian ; Luo, Cheng ; Luo, Xiao-min ; Chen, Shi-jie ; Wang, Yong-hui
Publisher:Singapore: Springer Singapore
Journal title:Acta pharmacologica Sinica, 2021-09, Vol.42 (9), p.1524-1534
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 13
ArticlesPeer ReviewedFull Text
Molecular Dynamics Simulations Based on 1-Phenyl-4-Benzoyl-1-Hydro-Triazole ERRα Inverse Agonists
Author / Creator:Gao, Zhipei ; Du, Yongli ; Sheng, Xiehuang ; Shen, Jingkang
Publisher:Switzerland: MDPI AG
Journal title:International journal of molecular sciences, 2021-04, Vol.22 (7), p.3724
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 14
ArticlesPeer ReviewedFull Text
Piperazine- and Piperidine-Containing Thiazolo[5,4-d]pyrimidine Derivatives as New Potent and Selective Adenosine A2A Receptor Inverse Agonists
Author / Creator:Varano, Flavia ; Catarzi, Daniela ; Vigiani, Erica ; Vincenzi, Fabrizio ; Pasquini, Silvia ; Varani, Katia ; Colotta, Vittoria
Publisher:Basel: MDPI AG
Journal title:Pharmaceuticals (Basel, Switzerland), 2020-07, Vol.13 (8), p.161
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 15
ArticlesPeer ReviewedFull Text
Flipping the GPCR Switch: Structure-Based Development of Selective Cannabinoid Receptor 2 Inverse Agonists
Author / Creator:Kosar, Miroslav ; Sarott, Roman C. ; Sykes, David A. ; Viray, Alexander E. G. ; Vitale, Rosa Maria ; Tomašević, Nataša ; Li, Xiaoting ; Ganzoni, Rudolf L. Z. ; Kicin, Bilal ; Reichert, Lisa ; Patej, Kacper J. ; Gómez-Bouzó, Uxía ; Guba, Wolfgang ; McCormick, Peter J. ; Hua, Tian ; Gruber, Christian W. ; Veprintsev, Dmitry B. ; Frank, James A. ; Grether, Uwe ; Carreira, Erick M.
Publisher:United States: American Chemical Society
Journal title:ACS central science, 2024-05, Vol.10 (5), p.956-968
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 16
ArticlesPeer ReviewedFull Text
RORγt inverse agonists demonstrating a margin between inhibition of IL-17A and thymocyte apoptosis RORγt inverse agonists demonstrating a margin between inhibition of IL-17A and thymocyte apoptosis
Author / Creator:Mia Collins ; Rikard Pehrson ; Hanna Grindebacke ; Agnes Leffler ; Marie Ramnegård ; Helena Rannikmäe ; Nina Krutrök ; Linda Yrlid ; Charlotte Pollard ; Ian Dainty ; Frank Narjes ; Stefan von Berg ; Antonio Llinas ; Anna Malmberg ; Jane McPheat ; Eva Hansson ; Elisabeth Bäck ; Jenny Bernström ; Thomas G. Hansson ; David Keeling ; Johan Jirholt
Publisher:Public Library of Science (PLoS)
Journal title:PloS one, 2025-01, Vol.20 (1)
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 17
ArticlesPeer ReviewedFull Text
Structure-Based Identification of Potent Natural Product Chemotypes as Cannabinoid Receptor 1 Inverse Agonists
Author / Creator:Pandey, Pankaj ; Roy, Kuldeep K. ; Liu, Haining ; Ma, Guoyi ; Pettaway, Sara ; Alsharif, Walid F. ; Gadepalli, Rama S. ; Rimoldi, John M. ; McCurdy, Christopher R. ; Cutler, Stephen J. ; Doerksen, Robert J.
Publisher:Switzerland: MDPI
Journal title:Molecules (Basel, Switzerland), 2018-10, Vol.23 (10), p.2630
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 18
ArticlesPeer ReviewedFull Text
Biology and therapeutic potential of cannabinoid CB2 receptor inverse agonists
Author / Creator:Lunn, C A ; Reich, E‐P ; Fine, J S ; Lavey, B ; Kozlowski, J A ; Hipkin, R W ; Lundell, D J ; Bober, L
Publisher:Oxford, UK: Blackwell Publishing Ltd
Journal title:British journal of pharmacology, 2008-01, Vol.153 (2), p.226-239
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 19
ArticlesPeer ReviewedFull Text
2-Arylpropionic Acid Pyrazolamides as Cannabinoid CB2 Receptor Inverse Agonists Endowed with Anti-Inflammatory Properties
Author / Creator:de Oliveira, Daniela R. ; Maia, Rodolfo C. ; de Carvalho França, Patrícia R. ; Fernandes, Patrícia D. ; Barbosa, Gisele ; Lima, Lídia M. ; Fraga, Carlos A. Manssour
Publisher:Switzerland: MDPI AG
Journal title:Pharmaceuticals (Basel, Switzerland), 2022-12, Vol.15 (12), p.1519
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.
Export this record
Export to excel
Print
Export record to excel
File type to download
Beta version
Select record 20
ArticlesPeer ReviewedFull Text
Docking 14 Million Virtual Isoquinuclidines against the μ and κ Opioid Receptors Reveals Dual Antagonists–Inverse Agonists with Reduced Withdrawal Effects
Author / Creator:Vigneron, Seth F. ; Ohno, Shohei ; Braz, Joao ; Kim, Joseph Y. ; Kweon, Oh Sang ; Webb, Chase ; Billesbølle, Christian B. ; Srinivasan, Karthik ; Bhardwaj, Karnika ; Irwin, John J. ; Manglik, Aashish ; Basbaum, Allan I. ; Ellman, Jonathan A. ; Shoichet, Brian K.
Publisher:United States: American Chemical Society
Journal title:ACS central science, 2025-05, Vol.11 (5), p.770-790
View online as a Library member
Access ebook if you are in the Library. Registered NSW residents may log in from home.

Showing 1 to 20 of 2,731 results

Export record to excel

Export this record

Export record to excel

Advanced fluorescence microscopy reveals disruption of dynamic CXCR4 dimerization by subpocket-specific inverse agonists

Export this record

Export record to excel

RO4938581, a novel cognitive enhancer acting at GABAA α5 subunit-containing receptors

Export this record

Export record to excel

RORγt inverse agonists demonstrating a margin between inhibition of IL-17A and thymocyte apoptosis

Export this record

Export record to excel

Structural mechanism of CB1R binding to peripheral and biased inverse agonists

Export this record

Export record to excel

β-Arrestin-Mediated Activation of MAPK by Inverse Agonists Reveals Distinct Active Conformations for G Protein-Coupled Receptors

Export this record

Export record to excel

ROR[gamma]t inverse agonists demonstrating a margin between inhibition of IL-17A and thymocyte apoptosis

Export this record

Export record to excel

Targeting Oxidative Stress: Novel Coumarin-Based Inverse Agonists of GPR55

Export this record

Export record to excel

Identification of Selective ERRγ Inverse Agonists

Export this record

Export record to excel

Identification of Selective ERR[gamma] Inverse Agonists

Export this record

Export record to excel

Towards Translation of PqsR Inverse Agonists: From In Vitro Efficacy Optimization to In Vivo Proof‐of‐Principle

Export this record

Export record to excel

The discovery of a novel series of potential ERRα inverse agonists based on p-nitrobenzenesulfonamide template for triple-negative breast cancer in vivo

Export this record

Export record to excel

Crystallography-guided discovery of carbazole-based retinoic acid-related orphan receptor gamma-t (RORγt) modulators: insights into different protein behaviors with “short” and “long” inverse agonists

Export this record

Export record to excel

Molecular Dynamics Simulations Based on 1-Phenyl-4-Benzoyl-1-Hydro-Triazole ERRα Inverse Agonists

Export this record

Export record to excel

Piperazine- and Piperidine-Containing Thiazolo[5,4-d]pyrimidine Derivatives as New Potent and Selective Adenosine A2A Receptor Inverse Agonists

Export this record

Export record to excel

Flipping the GPCR Switch: Structure-Based Development of Selective Cannabinoid Receptor 2 Inverse Agonists

Export this record

Export record to excel

RORγt inverse agonists demonstrating a margin between inhibition of IL-17A and thymocyte apoptosis RORγt inverse agonists demonstrating a margin between inhibition of IL-17A and thymocyte apoptosis

Export this record

Export record to excel

Structure-Based Identification of Potent Natural Product Chemotypes as Cannabinoid Receptor 1 Inverse Agonists

Export this record

Export record to excel

Biology and therapeutic potential of cannabinoid CB2 receptor inverse agonists

Export this record

Export record to excel

2-Arylpropionic Acid Pyrazolamides as Cannabinoid CB2 Receptor Inverse Agonists Endowed with Anti-Inflammatory Properties

Export this record

Export record to excel

Docking 14 Million Virtual Isoquinuclidines against the μ and κ Opioid Receptors Reveals Dual Antagonists–Inverse Agonists with Reduced Withdrawal Effects

Refine your search